LEGEND:
PRO means either an inactive drug which is metabolized to an active drug or is an (less) active drug which will be metabolized to another active metabolite.
SUB means a drug which is metabolized to an inactive metabolite.
INH is a drug which will increase the concentration of another drug.
IND is a drug which will decrease the concentration of another drug.
The different green colours means the intensity of a drug to be metabolized by its protein (enzyme/transporter), the grey means its intensity (=strength) and clinical relevance is unknown:
Unknown
Weak
Medium
Strong

Substance
Phase I - Enzymes (inactivate substrate, activate prodrug) Phase II - Conjugation Enzymes (make substrate water-soluble) Phase III - Drug Transport Proteins (affect absorption & excretion)
MAO Oxydation by Cytochrome P-450 (CYP) Oxydation by flavin-containing monooxygenase (FMO) Reduction Enzyme Glucuronidation by UDP-Glucuronosyltransferase (UGT) Acetylation Efflux-Transporter Solute-Carrier Transporter (SLCT) = Influx & Efflux transporter
MAO-A 1A2 2A6 2B6 2C8 2C9 3A5 2C19 2D6 2E1 3A4 FMO DPD VKORC1 1A1 1A3 1A4 1A6 1A9 2B4 2B7 2B10 2B15 2B17 NAT2 ABCG2 (BCRP) ABCB1 (Pgp,MDR) OAT1 OAT3 OCT2 MATE1 MATE-2K OATP1B3 SLCO1B1 (OATP1B1)
Abiraterone
Acenocoumarol
Acetaminophen (Paracetamol)
Acyclovir
Adefovir
Agomelatine
Alfentanil
Allopurinol
Alosetron
Alprazolam
Alprenolol
Amiodarone
Amitriptyline
Amlodipine
Amodiaquine
Apixaban
Aprepitant
Aripiprazole
Armodafinil
Artemether
Artemisinin
Astemizole
Asunaprevir
Atazanavir
Atomoxetine
Atorvastatin
Avanafil
Beta-Naphthoflavone
Bilirubin
Bisoprolol
Boceprevir
Bortezomib
Bosentan
Broccoli
Bromocriptine
Brussel Sprouts
Budesonide
Bufuralol
Buprenorphine
Bupropion
Buspirone
Caffeine
Cannabidiol
Carbamazepine
Carisoprodol
Carvedilol
Cefaclor
Ceftizoxime
Celecoxib
Celiprolol
Cerivastatin
Char-Grilled Meat
Chloramphenicol
Chloroquine
Chlorpheniramine
Chlorpromazine
Chlorzoxazone
Ciclosporin (Cyclosporine)
Cilostazol
Cimetidine
Cinacalcet
Ciprofibrate
Ciprofloxacin
Cisapride
Citalopram
Clarithromycin
Clemastine
Clobazam
Clomipramine
Clonazepam
Clonidine
Clopidogrel
Clotrimazole
Clozapine
Cobicistat
Cocaine
Codeine
Colchicine
Conivaptan
Cortisol
Crizotinib
Curcumin
Cyclobenzaprine
Cyclophosphamide
Dabigatran
Daclatasvir
Danoprevir
Dapsone
Darifenacin
Darunavir
Dasabuvir
Dasatinib
Debrisoquine
Deferasirox
Delavirdine
Desipramine
Desogestrel
Desvenlafaxine (active metabolite of venlafaxine)
Dexamethasone
Tenofovir
Dexfenfluramine
Dextromethorphan
Diazepam
Diclofenac
Dienogest
Diethyldithiocarbamate
Rivaroxaban
Dihydralazine
Dihydrocodeine
Dihydroergotamine
Diltiazem
Dimethylformamide
Diosmin
Diphenhydramine
Dipyridamole
Disulfiram
Docetaxel
Dofetilide
Dolutegravir
Domperidone
Donepezil
Doxepin
Doxorubicin (Adriamycin®)
Doxycycline
Dronedarone
Duloxetine
Dutasteride
Ebastine
Ecstasy (Mdma)
Efavirenz
Eletriptan
Eliglustat
Eltrombopag
Elvitegravir
Encainide
Enflurane
Enoxacin
Enzalutamide
Eplerenone
Ergotamine
Erlotinib
Erythromycin
Escitalopram (S-citalopram)
Esomeprazole
Estradiol
Ethanol
Ethinylestradiol
Ethosuximide
Etoposide
Etravirine
Everolimus
Famotidine
Felbamate
Felodipine
Fenofibrate
Fentanyl
Fexofenadine
Fibrate
Finasteride
Flecainide
Fluconazole
Fluoroquinolones
Fluorouracil (5-Fluorouracil)
Fluoxetine
Nortriptyline
Fluvastatin
Flurbiprofen
Fluvoxamine
Fosamprenavir
Fosaprepitant
Furafylline
Furosemide
Galantamine
Ganciclovir
Gefitinib
Gemfibrozil
Gestodene
Glibenclamide (Glyburide)
Gliclazide
Glimepiride
Glipizide
Glitazones
Glucocorticoids
Glyburide
Granisetron
Grapefruit
Halofantrine
Haloperidol
Halothane
Hexobarbital
Histamine H1 Receptor Antagonists
Hydrocodone
Hydrocortisone
Hydroxyzine
Hypericum (St. John's Wort)
Ibrutinib
Ibuprofen
Idelalisib
Ifosfamide
Imatinib
Imipramine
Indinavir
Indomethacin
Insulin
Interferon
Irbesartan
Irinotecan
Isoflurane
Isoniazid (isonicotinylhydrazide (INH))
Isradipine
Istradefylline
Itraconazole
Ivacaftor
Ketamine
Ketoconazole
Ketoprofen
Labetalol
Lamotrigin
Lansoprazole
Lapatinib
Ledipasvir
Lercanidipine
Letrozole
Levomepromazine
Lidocaine
Liquorice (licorice)
Lomitapide
Loperamide
Lopinavir
Lorazepam
Loratadine
Lorcaserin
Lornoxicam
Losartan
Lovastatin
Lumefantrine
Lurasidone
Maprotiline
Maraviroc
Medroxyprogesteron
Mefenamic Acid
Mefloquine
Melatonin
Meloxicam
Meperidine
Meprobamate
Mercaptopurin
Metamizole (Dipyrone)
Metformin
Methadone
Methotrexate
Methoxsalen (Xanthotoxin)
Methoxyflurane
Methylcholanthrene
Methylprednisolone
Metoclopramide
Metoprolol
Metronidazole
Mexiletine
Mianserine
Mibefradil
Miconazole
Midazolam
Midodrine
Mifepristone
Minaprine
Mirabegron
Mirtazapine
Mitotane
Moclobemide
Modafinil
Montelukast
Morphine
Mycophenolate Mofetil
Nabumetone
Nafcillin
Naloxegol
Naproxen
Nateglinide
Nebivolol
Nefazodone
Nelfinavir
Nevirapine
Nifedipine
Nilotinib
Nilutamide
Nimodipine
Nisoldipine
Nitrazepam
Nitrendipine
Norethindrone
Norethisterone
Norfloxacin
Norfluoxetine
Olanzapine
Ombitasvir
Omeprazole
Pantoprazole
Ondansetron
Oral Contraceptives
Oseltamivir
Oxazepam
Oxcarbazepine
Oxybutynine
Oxycodone
Paclitaxel
P-Aminohippuric Acid (Pah)
Paritaprevir
Paroxetine
Pazopanib
Peginterferon Alpha-2A
Penicillin G (Benzylpenicillin)
Perhexiline
Perphenazine
Phenacetin
Phenformin
Phenobarbital
Phenprocoumone
Phenylbutazone
Phenytoin
Pimozide
Pioglitazone
Piperine
Pirfenidone
Piroxicam
Pitavastatin
Posaconazole
Prasugrel
Pravastatin
Prednisolone
Prednisone
Primidone
Probenecid
Progesterone
Proguanil
Promethazine
Propafenone
Propofol
Propranolol
Quercetin
Quetiapine
Quinidine
Quinine
Rabeprazole
Ramelteon
Ramosetron
Ranitidine
Ranolazine
Reboxetine
Repaglinide
Rifabutin
Rifampin (Rifampicin)
Rilpivirine
Riluzole
Risperidone
Ritonavir
R-Mephobarbital
Romidepsin
Ropivacaine
Rosiglitazone
Rosuvastatin
Roxithromycine
Rufinamide
Salmeterol
Saquinavir
Saxagliptine
Secobarbital
Selegiline
Sertraline
Sevoflurane
Sildenafil
Silybum Marianum (milk thistle)
Simeprevir
Simvastatin
Sirolimus
S-Mephenytoin
Sofosbuvir
Sorafenib
Sparteine
Starfruit
Suboxone
Sufentanil
Sulfamethoxazole (SMZ, SMX)
Sulfaphenazole (sulfafenazol)
Sulfasalazine
Sunitinib
Suprofen
Tacrine
Tacrolimus
Tadalafil
Tamoxifen
Tamsulosine
Tasimelteon
Telaprevir
Telithromycin
Temsirolimus
Teniposide
Tenoxicam
Terbinafine
Terfenadine
Teriflunomide
Testosterone
Thc
Theophylline
Thioridazine
Thiotepa
Thyroxin (Levothyroxine)
Ticagrelor
Ticlopidine
Timolol
Tipranavir
Tizanidine
Tofisopam
Tolbutamide
Tolterodine
Tolvaptan
Topiramate
Torsemide (Torasemide)
Tramadol
Trazodone
Triamterene
Triazolam
Trimethoprim
Trimipramine
Tripelennamine
Troglitazone
Troleandomycin
Tropisetron
Valproic acid (valproate)
Vandetanib
Vardenafil
Vegetables
Vemurafenib
Venlafaxine
Verapamil
Vinblastine
Vincristine
Voriconazole
Warfarin
Zafirlukast
Zaleplon
Zileuton
Ziprasidone
Zolmitriptan
Zolpidem
Zopiclone
Zuclopenthixol
Tobacco smoke ( hydrocarbon, not nicotine)
Lamivudine
Raltegravir
Vinorelbine
Dacarbazine
Doravirine
Acetylsalicylic acid
Brivudin
Sorivudin
Candesartan
Digoxin
Azithromycin
Spironolactone
Hydrochlorothiazide
Abacavir
Fampridine
Acetaminophen (Paracetamol) toxic dose
Elbasvir
Grazoprevir
Hydralazine
Nicotine
Flupentixol
Melperon
Raloxifene
Fulvestrant
Cabergoline
Entacapone
Lisuride
Pergolide
Rasagiline
Biperiden
Ropinirole
Tolcapone
Clomethiazole
Hydroxychloroquine
Asenapin
Cyproterone
Amphetamine
Dextroamphetamine
Elexacaftor
Tezacaftor
remdesivir
Entrectinib
Siponimod
Gilteritinib
Ozanimod
Ropeginterferon alpha-2b
Darolutamid
Larotrectinib
Delafloxacine
Tucatinib
Alpelisib
Neratinib
Esketamin
Baloxavir
Lorlatinib
Upadacitinib
Apalutamid
Dacomitinib
Mercaptamine
Abemaciclib
Bictegravir
Emtricitabin
Natrium(4-phenylbutanoat)
Edaravone
Pitolisant
Selpercatinib
Ertugliflozin
Stiripentol
Brexpiprazol
Cariprazine
Venetoclax
Letermovir
Cabozantinib
Velpatasvir
Voxilaprevir
Isavuconazole
Glecaprevir
Baricitinib
Midostaurin
Lesinurad
Palbociclib
Alectinib
Ivermectin
Loxapin
Migalastat
Brivaracetam
Selexipag
Rizatriptane
Edoxaban
Opipramol
Tilidine
Nintedanib
nirmatrelvir
Hemin
Albendazole
Valsartan
Dapagliflozin
Formoterol
desloratadine
Help us to improve our table. If you think our table lacks a drug and/or a pharmacokinetic variable (info about CYP, UGT, efflux/uptake transporter), do not hesitate to inform us. After reviewed by our medical specialist for clinical pharmacology the information will be added to our table.